Gergely Makara: search on Z-Library

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1

Conformational analysis of a condensed macrocyclic β-lactam by NMR and molecular dynamics calculations

György M. Keseru&amp, #x030B, , Helga Vásárhelyi, Gergely Makara

Journal:

Journal of Molecular Structure

Year:

1994

Language:

english

File:

PDF, 329 KB

english, 1994

2

Synthesis of Bicyclic Pyrimidine Derivatives as ATP Analogues

Makara, Gergely M., Ewing, William, Ma, Yao, Wintner, Edward

Journal:

Journal of Organic Chemistry

Year:

2001

Language:

english

File:

PDF, 174 KB

english, 2001

3

A Single Vessel Protocol for the Efficient Formation of Amide Bonds from Esters and Lactones.

Noriyuki H. Kawahata, Jeseca Brookes, Gergely M. Makara

Journal:

Year:

2002

File:

PDF, 29 KB

2002

4

New Developments in Chemical Library Synthesis. Norbornenyl Tags for Use in Phase-Switching, Sequestration, Capture-Release and Soluble Support Applications

Daniel L. Flynn, Paul R. Hanson, Scott C. Berk, Gergely M. Makara

Journal:

Year:

2003

File:

PDF, 59 KB

2003

5

Recent Advances in Chemical Library Synthesis Methodology

Daniel L. Flynn, Scott C. Berk, Gergely M. Makara

Journal:

Year:

2003

File:

PDF, 50 KB

2003

6

Synthesis, molecular modeling, and evaluation of nonphenolic indole analogs of mycophenolic acid

Moustafa E El-Araby, Ralph J Bernacki, Gergely M Makara, Paula J Pera, Wayne K Anderson

Journal:

Bioorganic & Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 447 KB

english, 2004

7

Improving success rates for lead generation using affinity binding technologies

Gergely M Makara, John Athanasopoulos

Journal:

Current Opinion in Biotechnology

Year:

2005

Language:

english

File:

PDF, 259 KB

english, 2005

8

Activation of carboxylic acids by Burgess reagent: an efficient route to acyl ureas and amides

Derek Wodka, Michael Robbins, Ping Lan, Rogelio L. Martinez, John Athanasopoulos, Gergely M. Makara

Journal:

Tetrahedron Letters

Year:

2006

Language:

english

File:

PDF, 94 KB

english, 2006

9

An efficient method to access 2-substituted benzimidazoles under solvent-free conditions

Ping Lan, F. Anthony Romero, Threshia S. Malcolm, Benjamin D. Stevens, Dariusz Wodka, Gergely M. Makara

Journal:

Tetrahedron Letters

Year:

2008

Language:

english

File:

PDF, 141 KB

english, 2008

10

Michael addition of amines to vinyl sulfonamides on solid support

Gergely M Makara, Yao Ma

Journal:

Tetrahedron Letters

Year:

2001

Language:

english

File:

PDF, 81 KB

english, 2001

11

An efficient solid-phase synthesis of 3-alkylamino-1,2,4-oxadiazoles

Gergely M Makara, Peter Schell, Kelley Hanson, Dennis Moccia

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 95 KB

english, 2002

12

A single vessel protocol for the efficient formation of amide bonds from esters and lactones

Noriyuki H. Kawahata, Jeseca Brookes, Gergely M. Makara

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 170 KB

english, 2002

13

A facile synthesis of 3-substituted pipecolic acids, chimeric amino acids

Gergely M. Makara, Garland R. Marshall

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 247 KB

english, 1997

14

Bound conformations for ligands for G-protein coupled receptors

Garland R. Marshall, Rino Ragno, Gergely M. Makara, Rieko Arimoto, Oleg Kisselev

Journal:

International Journal of Peptide Research and Therapeutics

Year:

1999

Language:

english

File:

PDF, 642 KB

english, 1999

15

The influence of lead discovery strategies on the properties of drug candidates

Keserü, György M., Makara, Gergely M.

Journal:

Nature Reviews Drug Discovery

Year:

2009

Language:

english

File:

PDF, 454 KB

english, 2009

16

Bound conformations for ligands for G-protein coupled receptors

Garland R. Marshall, Rino Ragno, Gergely M. Makara, Rieko Arimoto, Oleg Kisselev

Journal:

International Journal of Peptide Research and Therapeutics

Year:

1999

Language:

english

File:

PDF, 96 KB

english, 1999

17

A reagent-based strategy for the design of large combinatorial libraries: A preliminary experimental validation

Gergely M. Makara, Huw Nash, Zhongli Zheng, Jean-Paul A. Orminati, Edward A. Wintner

Journal:

Molecular Diversity

Year:

2003

Language:

english

File:

PDF, 435 KB

english, 2003

18

Hit discovery and hit-to-lead approaches

György M. Keserű, Gergely M. Makara

Journal:

Drug Discovery Today

Year:

2006

Language:

english

File:

PDF, 243 KB

english, 2006

19

On the mechanism of the alkylation of quinoline and naphthyridine derivatives

Makara, Gergely, Keserű, György M., Kovács, Attila

Journal:

Journal of the Chemical Society Perkin Transactions 2

Year:

1994

Language:

english

File:

PDF, 536 KB

english, 1994

20

Rhodopsin-Transducin Interface: Studies with Conformationally Constrained Peptides

Arimoto, Rieko, Kisselev, Oleg G., Makara, Gergely M., Marshall, Garland R.

Journal:

Biophysical Journal

Year:

2001

Language:

english

File:

PDF, 326 KB

english, 2001

21

On the Conformation of Tiazofurin Analogues

Makara, Gergely M., Keserû, György M.

Journal:

Journal of Medicinal Chemistry

Year:

1997

Language:

english

File:

PDF, 436 KB

english, 1997

22

Combinatorial Synthesis of Substituted Biaryls and Heterocyclic Arylamines

Ma, Yao, Margarida, Laura, Brookes, Jeseca, Makara, Gergely M., Berk, Scott C.

Journal:

Journal of Combinatorial Chemistry

Year:

2004

Language:

english

File:

PDF, 74 KB

english, 2004

23

On Sampling of Fragment Space

Makara, Gergely M.

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 136 KB

english, 2007

24

Solid-Phase Synthesis of 3-Alkylamino-1,2,4-triazoles

Makara, Gergely M., Ma, Yao, Margarida, Laura

Journal:

Organic Letters

Year:

2002

Language:

english

File:

PDF, 52 KB

english, 2002

25

Measuring Molecular Similarity and Diversity: Total Pharmacophore Diversity

Makara, Gergely M.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 543 KB

english, 2001

26

Versatile Solid-Phase Synthesis of Trisubstituted 1 H -Pyrido[2,3- d ]pyrimidin-4-ones and Related Heterocycles

Schell, Peter, Richards, Matthew P., Hanson, Kelley, Berk, Scott C., Makara, Gergely M.

Journal:

Journal of Combinatorial Chemistry

Year:

2005

Language:

english

File:

PDF, 102 KB

english, 2005

27

Nuclear Magnetic Resonance and Molecular Modeling Study on Mycophenolic Acid: Implications for Binding to Inosine Monophosphate Dehydrogenase

Makara, Gergely M., Keserû, György M., Kajtár-Peredy, Mária, Anderson, Wayne K.

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 214 KB

english, 1996

28

Synthesis and Modeling Studies with Monocyclic Analogues of Mycophenolic Acid

Anderson, Wayne K., Boehm, Terri L., Makara, Gergely M., Swann, R. Thomas

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 345 KB

english, 1996

29

An Efficient Synthesis of 5,7-Dimethoxy-4-methylphthalide, a Key Intermediate in the Synthesis of Mycophenolic Acid

Makara, Gergely M., Anderson, Wayne K.

Journal:

Journal of Organic Chemistry

Year:

1995

Language:

english

File:

PDF, 280 KB

english, 1995

30

An Improved Synthesis of 5,7-Dimethoxy-4-methylphthalide, A Key Intermediate in the Synthesis of Mycophenolic Acid

Makara, Gergely M., Klubek, Kevin, Anderson, Wayne K.

Journal:

Synthetic Communications

Year:

1996

Language:

english

File:

PDF, 268 KB

english, 1996

31

Label-Free High-Throughput Screening via Mass Spectrometry: A Single Cystathionine Quantitative Method for Multiple Applications

Holt, Tom G., Choi, Bernard K., Geoghagen, Neil S., Jensen, Kristian K., Luo, Qi, LaMarr, William A., Makara, Gergely M., Malkowitz, Lorraine, Ozbal, Can C., Xiong, Yusheng, Dufresne, Claude, Luo, Min

Journal:

Assay and Drug Development Technologies

Year:

2009

Language:

english

File:

PDF, 1.10 MB

english, 2009

32

Synthesis of Condensed Heterocycles by the Gould–Jacobs Reaction in a Novel Three-Mode Pyrolysis Reactor

Lengyel, László Csaba, Sipos, Gellért, Sipőcz, Tamás, Vágó, Teréz, Dormán, György, Gerencsér, János, Makara, Gergely, Darvas, Ferenc

Journal:

Organic Process Research & Development

Year:

2015

Language:

english

File:

PDF, 1.02 MB

english, 2015

33

Predictive value of psychosocial assessment for the mortality of patients waiting for liver transplantation

Gazdag, Gábor, Horváth, G Gergely, Makara, Mihály, Ungvari, Gabor S, Gerlei, Zsuzsanna

Journal:

Psychology Health & Medicine

Year:

2015

Language:

english

File:

PDF, 537 KB

english, 2015

34

ChemInform Abstract: Synthesis of Condensed Heterocycles by the Gould-Jacobs Reaction in a Novel Three-Mode Pyrolysis Reactor.

Lengyel, Laszlo Csaba, Sipos, Gellert, Sipocz, Tamas, Vago, Terez, Dorman, Gyoergy, Gerencser, Janos, Makara, Gergely, Darvas, Ferenc

Journal:

Year:

2015

File:

PDF, 25 KB

2015

35

Effect of hepatitis C infection on the quality of life

Horváth, Gergely, Keleti, Teodóra, Makara, Mihály, Ungvari, Gabor S., Gazdag, Gábor

Journal:

Perspectives In Psychiatric Care

Year:

2018

Language:

english

File:

PDF, 175 KB

english, 2018